問題詳情

30 Thioperamide 可以較具選擇性的拮抗下列何種受體的作用?
(A) 5-HT 2
(B)H 2
(C) 5-HT 3
(D)H 3

參考答案

答案:D
難度:困難0.394886
統計:A(150),B(78),C(198),D(278),E(0)

用户評論

Jason】評論

Histamine作用在H3受器上可抑制histamine之釋放,而H3受器拮抗劑 thioperamide可使histamine釋放出來而達到減少食物的攝取效果,但此效果會被H1受器拮抗劑 chlorpheniramine所阻斷。

郭蓉】評論

This receptor has been proposed as a target for treating sleep disorders.[9] The receptor has also been proposed as a target for treating neuropathic pain.[10]Because of its ability to modulate other neurotransmitters, H3 receptor ligands are being investigated for the treatment of numerous neurological conditions, including obesity (because of the histamine/orexinergic system interaction), movement disorders (because of H3 receptor-modulation of dopamine and GABA in the basal ganglia), schizophrenia and ADHD (again because of dopamine modulation) and research is underway to d...

張詠婷】評論

23 下列那一種藥物是Histamine H 3 receptors 的拮抗劑? (A)Thioperamide (B)α-methylhistamine (C)Imetit (D)Immepip 編輯私有筆記及自訂標籤

麻糬好好吃】評論

H3 agonist  ★★★★★★☆-☆☆☆☆☆-...