問題詳情

12.下列何者與theophylline併用時,會增加theophylline的代謝?
(A)phenytoin
(B)erythromycin
(C)ciprofloxacin
(D)cimetidine

參考答案

答案:A
難度:簡單0.8
書單:沒有書單,新增

用户評論

滾筒洗衣機】評論

theophylline為1A2及3A4受質p-gp +CYP廣誘導劑 : ET(E : 抗癲癇、T : 結核病);CYP3A4及p-gp強效通打phenytoinCYP1A2 (weak), CYP3A4 (strong)carbamazepineCYP1A2 (weak), CYP2C9 (weak), CYP3A4 (strong),phenobarbitalCYP1A2 (weak), CYP2C9 (weak), CYP3A4 (strong)RifampinCYP1A2 (weak), CYP2C19 (strong), CYP2C9 (moderate), CYP3A4 (strong)St. John's wortCYP3A4 (strong)--------------------------------------------------------------------------------------------------------------------CYP3A4強抑制劑 : MAC (M : macrolide、A : -azole、C : non-DHP CCB)Macrolide除了azithromycinAzolefluconazole, itraconazolenon...

加賴叫過去】評論

Theophylline大補帖來囉...

吳富豪】評論

CYP1A2受質誘★★★★★...

強力施巴】評論

Therapeutic range : 5-15 ug/ml (peak)