問題詳情

76 下列有關 vigabatrin 的敘述,何者錯誤?
(A)為 GABA 的結構類似物
(B)具有抑制 GABA 轉胺酶(transaminase)的活性
(C)適用於治療局部性癲癇及 West’s syndrome
(D)其 R(-)化學異構物為主要的有效成分

參考答案

答案:D
難度:簡單0.774648
統計:A(4),B(8),C(4),D(55),E(0)

用户評論

【用戶】Bryan

【年級】國三上

【評論內容】Drug Classes → Central Nervous System Agents → Anticonvulsants → Gamma-aminobutyric Acid Analogs : vigabatrin Gamma-aminobutyric acid (GABA) analogs are drugs that are similar to gamma-aminobutyric acid neurotransmitter, which is an inhibitory neurotransmitter. These analogs act as GABA-B receptors agonists and cause inhibitory action like GABA.

【用戶】Bryan

【年級】國三上

【評論內容】(D)其 S(+)enantiomer化學異構物為主要的有效成分

【用戶】Bryan

【年級】國三上

【評論內容】(D)其 S(+)enantio.....看完整詳解

【用戶】Bryan

【年級】國三上

【評論內容】Drug Classes → Central Nervous System Agents → Anticonvulsants → Gamma-aminobutyric Acid Analogs : vigabatrin Gamma-aminobutyric acid (GABA) analogs are drugs that are similar to gamma-aminobutyric acid neurotransmitter, which is an inhibitory neurotransmitter. These analogs act as GABA-B receptors agonists and cause inhibitory action like GABA.