【小羊】評論
Nicotinic receptor:Na+, K+M1,3,5 receptor: GqM2,4 receptor: Gi GABAA receptor:Cl-GABAB receptor:Gi 5-HT3 receptor:Na+, K+5-HT1 receptor:Gi5-HT2 receptor:Gq5-HT4 receptor:Gs NMDA receptor: Ca2+,Na+, K+AMPA receptor: Na+Kainate receptor: K+,Na+Glycine receptor: Cl- α1 receptor: Gqα2 receptor: Giβ1,β2 receptor: GsH1 receptor:GqH2 receptor:GsOpioid receptor: G...
【王瑜】評論
Lamotrigine:作用於電位敏感的鈉通道,安定神經膜及抑制興奮性氨基酸 (Glutamate)的釋放。
【滴水之恩湧泉以報】評論
前人大神整理NMDA:Na、Ca、K,興奮型⊖NMDA 藥物:1. Amantadine:治療帕金森2. Memantine:治療阿茲海默症3. Ketamine、Phencyclidine (PCP):神經興奮劑,解離型麻醉4. Felbamate:難治療的癲癇,有再生不良貧血、體重下降的副作用5. Lomotrigine:癲癇以下四個受器依受體亞型不同分屬於IR與GPCR, 而IR受體亞型以表格中四個為主 離子通道受器亞型(IR) 口訣 離婚海人早晚飯前三根菸TypeSubtypeEndogenous LigandGlutamateKainate(海人草酸) /AMPA(早上晚上)/ NMDAGlutamateGABAA/C (飯前)GABA(Cl-)Serotonine5HT-3 (三根)5-HTAcetylchlorideNicotine(菸鹼)AchSubstrateGPCR (Gq)GPCR(Gs)GPCR(Gi)Ligand gatedIon channelNE, Epiα...
【所得皆所愿】評論
Iontropic Receptor 離子通道型接受器Nicotine receptorAChNa+GABAA receptorGABACl-5-HT3SerotoninNa+ K+NMDA receptorGlutamic acidNa+AMPA receptorGlutamic acidNa+ K+ Ca2+
【過過小藥師】評論
Gt→cGMP視覺:Photons、Rhodopsin(視紫紅質)Golf→AC, cAMP↑嗅覺:odorantsGs→AC, cAMP↑β全部D1,5H2、V25-HT4PGI2ACTH(促腎上腺皮質素)Glucagon(升糖素)PTH(副甲狀腺素)TSH(促甲狀腺激素)Gi→AC, cAMP↓→K+↑α2, M2,AT-2偶數D2,3,4 5-HT1GABAB(肌肉鬆弛)OpioidsGq→PLC, IP3, DAG, Ca2+↑(PLC會將PIP2分解成IP3和DAG,然後IP3會活化Ca2+通道使Ca2+↑)α1, M1,AT-1奇數 H1、V15-HT2 ...